PMA也称TPA,全称为Phorbol-12-myristate-13-acetate (PMA),或12-O-Tetradecanoylphorbol 13-acetate(TPA),是一种最常用的佛波酯(phorbol ester)。PMA可以结合PKC,并激活PKC,随后导致一系列的细胞响应。PMA可以抑制Fas诱导的细胞凋亡,但又可以诱导HL-60细胞的凋亡。PMA在肝细胞中可以诱导iNOS的表达。PMA可以增强forskolin诱导的cAMP形成。PMA是一种促瘤剂,可以促进小鼠皮肤的成瘤。
PMA的分子量为616.84,分子式为C36H56O8,CAS Number:16561-29-8。本产品纯度大于99%。
本产品为进口分装,其中10mg/ml包装产品用DMSO配制,共0.1ml。5mg包装为粉末装。
包装清单:
产品编号 | 产品名称 | 包装 |
S1819-1mg | PMA/TPA (PKC激活剂) | 10mg/ml×0.1ml |
S1819-5mg | PMA/TPA (PKC激活剂) | 5mg |
S1819-25mg | PMA/TPA (PKC激活剂) | 25mg |
— | 说明书 | 1份 |
保存条件:
-20℃避光保存,半年有效。
注意事项:
本产品对人体有刺激性,操作时请小心,并注意适当防护以避免直接接触人体或吸入体内。
本产品在4℃、冰浴等较低温度情况下会凝固而粘在离心管管底、管壁或管盖内,可以20-25℃水浴温育片刻至全部融解后使用。
本产品仅限于专业人员的科学研究用,不得用于临床诊断或治疗,不得用于食品或药品,不得存放于普通住宅内。
为了您的安全和健康,请穿实验服并戴一次性手套操作。
使用说明:
1. PMA常见使用浓度范围为0.1-10μM,最常见的使用浓度为1μM。具体的最佳工作浓度请参考相关文献,或根据实验目的,以及所培养的特定细胞和组织,通过实验进行摸索和优化。
产品编号
|
产品名称
|
产品包装
|
S1563
|
Cyclosporin A
(免疫抑制剂/PP2B抑制剂)
|
50mg
|
S1612-1mg
|
Forskolin (腺苷酸环化酶激活剂)
|
5mg/ml×0.2ml
|
S1612-5mg
|
Forskolin (腺苷酸环化酶激活剂)
|
5mg
|
S1612-25mg
|
Forskolin (腺苷酸环化酶激活剂)
|
25mg
|
S1672-250nmol
|
Ionomycin (钙离子载体)
|
5mM×0.05ml
|
S1672-1μmol
|
Ionomycin (钙离子载体)
|
5mM×0.2ml
|
S1672-5mg
|
Ionomycin (钙离子载体)
|
5mg
|
S1819-1mg
|
PMA/TPA (PKC激活剂)
|
10mg/ml×0.1ml
|
S1819-5mg
|
PMA/TPA (PKC激活剂)
|
5mg
|
S1819-25mg
|
PMA/TPA (PKC激活剂)
|
25mg
|
S1882
|
Staurosporine
(PKC抑制剂)
|
0.1mg
|
S1883
|
Staurosporine
(PKC抑制剂)
|
0.5mg
|
S1888
|
Trequinsin (PDE
III抑制剂)
|
2mg
|
SD0011-10mM
|
Endoxifen HCl
(Estrigen Receptor拮抗剂)
|
10mM
|
SD0011-5mg
|
Endoxifen HCl
(Estrigen Receptor拮抗剂)
|
5mg
|
SD0011-25mg
|
Endoxifen HCl
(Estrigen Receptor拮抗剂)
|
25mg
|
SD2371-10mM
|
Rimonabant
(Cannabinoid Receptor拮抗剂)
|
10mM
|
SD2371-5mg
|
Rimonabant
(Cannabinoid Receptor拮抗剂)
|
5mg
|
SD2371-25mg
|
Rimonabant
(Cannabinoid Receptor拮抗剂)
|
25mg
|
SD2375-10mM
|
AM251 (Cannabinoid
Receptor拮抗剂)
|
10mM
|
SD2375-5mg
|
AM251 (Cannabinoid
Receptor拮抗剂)
|
5mg
|
SD2375-25mg
|
AM251 (Cannabinoid
Receptor拮抗剂)
|
25mg
|
SD2380-10mM
|
Plerixafor (CXCR抑制剂)
|
10mM
|
SD2380-5mg
|
Plerixafor (CXCR抑制剂)
|
5mg
|
SD2380-25mg
|
Plerixafor (CXCR抑制剂)
|
25mg
|
SD2384-10mM
|
TGR5 (GPCR19激动剂)
|
10mM
|
SD2384-5mg
|
TGR5 (GPCR19激动剂)
|
5mg
|
SD2384-25mg
|
TGR5 (GPCR19激动剂)
|
25mg
|
SD2393-10mM
|
S1RA (Sigma
Receptor拮抗剂)
|
10mM
|
SD2393-5mg
|
S1RA (Sigma
Receptor拮抗剂)
|
5mg
|
SD2393-25mg
|
S1RA (Sigma
Receptor拮抗剂)
|
25mg
|
SD2398-10mM
|
MK-571 (LTD4受体拮抗剂)
|
10mM
|
SD2398-5mg
|
MK-571 (LTD4受体拮抗剂)
|
5mg
|
SD2398-25mg
|
MK-571 (LTD4受体拮抗剂)
|
25mg
|
SD2407-10mM
|
ZM241385 (Adenosine
Receptor抑制剂)
|
10mM
|
SD2407-5mg
|
ZM241385 (Adenosine
Receptor抑制剂)
|
5mg
|
SD2407-25mg
|
ZM241385 (Adenosine
Receptor抑制剂)
|
25mg
|
SD2420-10mM
|
Regadenoson
(Adenosine Receptor激动剂)
|
10mM
|
SD2420-5mg
|
Regadenoson
(Adenosine Receptor激动剂)
|
5mg
|
SD2420-25mg
|
Regadenoson
(Adenosine Receptor激动剂)
|
25mg
|
SD2429-10mM
|
AM630 (CB2拮抗剂)
|
10mM
|
SD2429-5mg
|
AM630 (CB2拮抗剂)
|
5mg
|
SD2429-25mg
|
AM630 (CB2拮抗剂)
|
25mg
|
SD2434-10mM
|
SCH58261 (Adenosine
Receptor抑制剂)
|
10mM
|
SD2434-5mg
|
SCH58261 (Adenosine
Receptor抑制剂)
|
5mg
|
SD2434-25mg
|
SCH58261 (Adenosine
Receptor抑制剂)
|
25mg
|
SD2438-10mM
|
SB334867 (OX
Receptor拮抗剂)
|
10mM
|
SD2438-5mg
|
SB334867 (OX
Receptor拮抗剂)
|
5mg
|
SD2438-25mg
|
SB334867 (OX
Receptor拮抗剂)
|
25mg
|
SD2443-10mM
|
Vilanterol (β2激动剂)
|
10mM
|
SD2443-5mg
|
Vilanterol (β2激动剂)
|
5mg
|
SD2443-25mg
|
Vilanterol (β2激动剂)
|
25mg
|
SD2447-10mM
|
Macitentan
(Endothelin Receptor拮抗剂)
|
10mM
|
SD2447-5mg
|
Macitentan
(Endothelin Receptor拮抗剂)
|
5mg
|
SD2447-25mg
|
Macitentan
(Endothelin Receptor拮抗剂)
|
25mg
|
SD2452-10mM
|
Vilazodone (SSRI抑制剂)
|
10mM
|
SD2452-5mg
|
Vilazodone (SSRI抑制剂)
|
5mg
|
SD2452-25mg
|
Vilazodone (SSRI抑制剂)
|
25mg
|
SD2465-10mM
|
AM281 (CB1拮抗剂)
|
10mM
|
SD2465-5mg
|
AM281 (CB1拮抗剂)
|
5mg
|
SD2465-25mg
|
AM281 (CB1拮抗剂)
|
25mg
|
SD2474-10mM
|
Reversine (Adenosine
Receptor拮抗剂)
|
10mM
|
SD2474-5mg
|
Reversine (Adenosine
Receptor拮抗剂)
|
5mg
|
SD2474-25mg
|
Reversine (Adenosine
Receptor拮抗剂)
|
25mg
|
SD2479-10mM
|
Umeclidinium
(mAChR抑制剂)
|
10mM
|
SD2479-5mg
|
Umeclidinium
(mAChR抑制剂)
|
5mg
|
SD2479-25mg
|
Umeclidinium
(mAChR抑制剂)
|
25mg
|
SD0006-10mM
|
PD123319 (RAAS抑制剂)
|
10mM
|
SD0006-25mg
|
PD123319 (RAAS抑制剂)
|
25mg
|
SD0006-5mg
|
PD123319 (RAAS抑制剂)
|
5mg
|
SD0015-10mM
|
LCZ696 (RAAS抑制剂)
|
10mM
|
SD0015-25mg
|
LCZ696 (RAAS抑制剂)
|
25mg
|
SD0015-5mg
|
LCZ696 (RAAS抑制剂)
|
5mg
|
SD0024-10mM
|
Azilsartan (RAAS拮抗剂)
|
10mM
|
SD0024-25mg
|
Azilsartan (RAAS拮抗剂)
|
25mg
|
SD0024-5mg
|
Azilsartan (RAAS拮抗剂)
|
5mg
|
SD3699-10mM
|
ZK811752 (CCR1拮抗剂)
|
10mM
|
SD3699-25mg
|
ZK811752 (CCR1拮抗剂)
|
25mg
|
SD3699-5mg
|
ZK811752 (CCR1拮抗剂)
|
5mg
|
SD9527-10mM
|
WAY100635 (5-HT1A拮抗剂)
|
10mM
|
SD9527-25mg
|
WAY100635 (5-HT1A拮抗剂)
|
25mg
|
SD9527-5mg
|
WAY100635 (5-HT1A拮抗剂)
|
5mg
|
SD9540-10mM
|
BMY7378 (5-HT
Receptor拮抗剂)
|
10mM
|
SD9540-25mg
|
BMY7378 (5-HT
Receptor拮抗剂)
|
25mg
|
SD9540-5mg
|
BMY7378 (5-HT
Receptor拮抗剂)
|
5mg
|
SD9549-10mM
|
JNJ-7777120
(Histamine Receptor拮抗剂)
|
10mM
|
SD9549-25mg
|
JNJ-7777120
(Histamine Receptor拮抗剂)
|
25mg
|
SD9549-5mg
|
JNJ-7777120
(Histamine Receptor拮抗剂)
|
5mg
|
SD9563-10mM
|
Brexpiprazole
(Dopamine Receptor激动剂)
|
10mM
|
SD9563-25mg
|
Brexpiprazole
(Dopamine Receptor激动剂)
|
25mg
|
SD9563-5mg
|
Brexpiprazole
(Dopamine Receptor激动剂)
|
5mg
|
SF6804-10mM
|
Vismodegib
(Hedgehog/Smoothened抑制剂)
|
10mM
|
SF6804-25mg
|
Vismodegib
(Hedgehog/Smoothened抑制剂)
|
25mg
|
SF6804-5mg
|
Vismodegib
(Hedgehog/Smoothened抑制剂)
|
5mg
|
SF6809-10mM
|
SANT-1
(Hedgehog/Smoothened拮抗剂)
|
10mM
|
SF6809-25mg
|
SANT-1
(Hedgehog/Smoothened拮抗剂)
|
25mg
|
SF6809-5mg
|
SANT-1
(Hedgehog/Smoothened拮抗剂)
|
5mg
|
SF2789-25mg
|
GSK690693 (Akt抑制剂)
|
25mg
|
SF2802-10mM
|
TGX221 (PI3K抑制剂)
|
10mM
|
SF2802-5mg
|
TGX221 (PI3K抑制剂)
|
5mg
|
SF2802-25mg
|
TGX221 (PI3K抑制剂)
|
25mg
|
SF2811-10mM
|
GSK2126458 (PI3K抑制剂)
|
10mM
|
SF2811-5mg
|
GSK2126458 (PI3K抑制剂)
|
5mg
|
SF2811-25mg
|
GSK2126458 (PI3K抑制剂)
|
25mg
|
SF2820-10mM
|
AZD5363 (Akt抑制剂)
|
10mM
|
SF2820-5mg
|
AZD5363 (Akt抑制剂)
|
5mg
|
SF2820-25mg
|
AZD5363 (Akt抑制剂)
|
25mg
|
SF2825-10mM
|
GSK2141795 (Akt抑制剂)
|
10mM
|
SF2825-5mg
|
GSK2141795 (Akt抑制剂)
|
5mg
|
SF2825-25mg
|
GSK2141795 (Akt抑制剂)
|
25mg
|
SF5337-10mM
|
R428 (Axl抑制剂)
|
10mM
|
SF5337-5mg
|
R428 (Axl抑制剂)
|
5mg
|
SF5337-25mg
|
R428 (Axl抑制剂)
|
25mg
|
SF5359-10mM
|
Masitinib (c-Kit抑制剂)
|
10mM
|
SF5359-5mg
|
Masitinib (c-Kit抑制剂)
|
5mg
|
SF5359-25mg
|
Masitinib (c-Kit抑制剂)
|
25mg
|
SF5422-10mM
|
Amuvatinib (c-Kit抑制剂)
|
10mM
|
SF5422-5mg
|
Amuvatinib (c-Kit抑制剂)
|
5mg
|
SF5422-25mg
|
Amuvatinib (c-Kit抑制剂)
|
25mg
|